SCHEMBL6158938

SCHEMBL6158938

CCCN1C(=O)CCC(NC(=O)c2cc(Cl)c(O)c(Cl)c2)C(=O)N1CC(=O)N(OCc1ccccc1)C1COC(=O)C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MME P08473 3/20 0.43
ACE P12821 3/20 0.43
RIPK1 Q13546 6/20 0.33
XIAP P98170 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
HSD17B13 Q7Z5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159304 0.90 MME (0.39) MMEACERIPK1XIAPKDM4E
SCHEMBL7668014 0.83 CCR2 (0.33) MMEACERIPK1
SCHEMBL6161334 0.82 MME (0.34) MMEACERIPK1XIAPTAS1R3
SCHEMBL6158934 0.79 MME (0.44) MMEACE
SCHEMBL6159042 0.74 KDM4E (0.33) KDM4EALDH1A1HPGD
SCHEMBL6159297 0.70 MME (0.40) MMEACERIPK1
SCHEMBL6158713 0.68 CASP1 (0.44) MMEACE
SCHEMBL6159420 0.66 XIAP (0.38) MMEACEXIAP
SCHEMBL5903274 0.66 CASP1 (0.54) RIPK1
SCHEMBL5903611 0.65 CASP1 (0.49) RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1062210-B1 1,2-DIAZEPANE DERIVATIVES AS INTERLEUKIN-1BETA CONVERTING ENZYME INHIBITORS VERTEX PHARMA (US) 2005-06-01 EP disclosed
US-6426413-B1 SUCH AS (N-BENZYLOXYCARBONYL-HYDRAZINO)-ACETIC ACID TERT-BUTYL ESTER; FOR PREVENTING AND TREATING INTERLEUKIN-MEDIATED DISEASES, APOPTOSIS, AUTOIMMUNE DISEASES, BONE DISORDERS, PROLIFERATIVE DISORDERS, INFECTIONS, AND DEGENERATIVE DISEASES VERTEX PHARMACEUTICALS INCORPORATED 2002-07-30 US disclosed