SCHEMBL7668014

SCHEMBL7668014

CS(=O)(=O)N1CCCC(NC(=O)c2cc(Cl)c(O)c(Cl)c2)C(=O)N1CC(=O)N(OCc1ccccc1)C1COC(=O)C1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.33
TERF2 Q15554 8/20 0.33
MME P08473 1/20 0.32
ACE P12821 1/20 0.32
CASP1 P29466 2/20 0.32
CASP8 Q14790 2/20 0.32
PLG P00747 1/20 0.32
PRSS1 P07477 1/20 0.32
TPSAB1 Q15661 1/20 0.32
TPSD1 Q9BZJ3 1/20 0.32
TPSG1 Q9NRR2 1/20 0.32
CASP3 P42574 1/20 0.32
RIPK1 Q13546 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159042 0.90 KDM4E (0.33) CCR2TERF2
SCHEMBL6158938 0.83 MME (0.43) MMEACERIPK1
SCHEMBL7668008 0.79 CASP3 (0.43) CASP1CASP8CASP3
SCHEMBL6161334 0.75 MME (0.34) MMEACERIPK1
SCHEMBL6159304 0.74 MME (0.39) MMEACERIPK1
SCHEMBL6159038 0.70 CASP3 (0.39) CASP1CASP8CASP3
SCHEMBL6160332 0.69 CASP1 (0.43) CASP1CASP8CASP3
SCHEMBL5903385 0.63 CASP1 (0.55) CASP1CASP8
SCHEMBL5903611 0.63 CASP1 (0.49) CASP1CASP8CASP3RIPK1
SCHEMBL3269454 0.63 KLK7 (0.53) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6426413-B1 SUCH AS (N-BENZYLOXYCARBONYL-HYDRAZINO)-ACETIC ACID TERT-BUTYL ESTER; FOR PREVENTING AND TREATING INTERLEUKIN-MEDIATED DISEASES, APOPTOSIS, AUTOIMMUNE DISEASES, BONE DISORDERS, PROLIFERATIVE DISORDERS, INFECTIONS, AND DEGENERATIVE DISEASES VERTEX PHARMACEUTICALS INCORPORATED 2002-07-30 US disclosed