SCHEMBL6162407

SCHEMBL6162407

Oc1ccc2nccc(Cl)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.50
ESR2 Q92731 3/20 0.50
ESRRB O95718 1/20 0.50
ESRRA P11474 1/20 0.50
TTR P02766 2/20 0.45
PARP1 P09874 1/20 0.44
MAPKAPK2 P49137 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
NR4A2 P43354 1/20 0.43
HSD17B10 Q99714 2/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 3/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
AXL P30530 1/20 0.41
PRKCI P41743 1/20 0.41
MAPT P10636 4/20 0.41
GAA P10253 2/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29729491 1.00 ESR1 (0.50) ESR1ESR2ESRRBESRRATTR
Bromide SCHEMBL9069911 0.98 ESR1 (0.49) ESR1ESR2ESRRBESRRATTR
SCHEMBL1043161 0.84 TLR8 (0.51) ESR1ESR2ESRRBESRRATTR
SCHEMBL29612575 0.84 TLR8 (0.51) ESR1ESR2ESRRBESRRATTR
Ammonia Solution, Strong SCHEMBL27616951 0.82 TLR8 (0.50) ESR1ESR2ESRRBESRRATTR
SCHEMBL1888577 0.79 NR4A2 (0.66) PARP1DYRK1BNR4A2HSD17B10MEN1
SCHEMBL30051309 0.79 NR4A2 (0.66) PARP1DYRK1BNR4A2HSD17B10MEN1
SCHEMBL30819181 0.79 PARP1 (0.47) PARP1MAPKAPK2NR4A2HSD17B10MEN1
SCHEMBL1332713 0.79 PARP1 (0.47) PARP1MAPKAPK2NR4A2HSD17B10MEN1
SCHEMBL29576809 0.78 TLR8 (0.43) DYRK1BNR4A2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260132121-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS INC (US) 2026-05-14 US disclosed
US-12624018-B1 Inhibitors of RIPK2 and medical uses thereof ODYSSEY THERAPEUTICS, INC. (US) 2026-05-12 US disclosed
US-12528791-B2 Thyroid hormone receptor beta agonist compounds TERNS PHARMACEUTICALS, INC. (US) 2026-01-20 US disclosed
US-20250319214-A1 A NOVEL KIT FOR RADIOPHARMACEUTICAL PREPARATION OF A RADIOMETAL LABELED CHELATE-FUNCTIONALIZED TARGETING CONJUGATE Life Molecular Imaging Ltd. (GB) 2025-10-16 US disclosed
EP-4622970-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2025-10-01 EP disclosed
WO-2024112854-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2024-05-30 WO disclosed
WO-2024112854-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2024-05-30 WO disclosed
WO-2023275195-A2 A NOVEL KIT FOR RADIOPHARMACEUTICAL PREPARATION OF A RADIOMETAL LABELED CHELATE-FUNCTIONALIZED TARGETING CONJUGATE LIFE MOLECULAR IMAGING LIMITED (GB) 2023-01-05 WO disclosed
US-20220281849-A1 THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS TERNS PHARMACEUTICALS, INC. 2022-09-08 US disclosed
EP-4017875-A1 THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS Terns Pharmaceuticals, Inc. (US) 2022-06-29 EP disclosed
CN-1181059-C Quinoline-4-base deviative I - 2004-12-22 CN disclosed
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US disclosed
US-6339093-B1 Isoquinoline derivatives HOFFMANN-LA ROCHE INC. 2002-01-15 US disclosed
EP-1090917-A1 Quinolin-4-yl derivatives and their use as NMDA-receptor subtype blockers F. HOFFMANN-LA ROCHE AG (CH) 2001-04-11 EP disclosed
CN-1290698-A Quinoline-4-base deviative I HOFFMANN LA ROCHE (CH) 2001-04-11 CN disclosed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP disclosed
US-5506235-A Quinoline derivatives as immunostimulants PFIZER INC. (US) 1996-04-09 US disclosed
EP-0597003-A1 QUINOLINE DERIVATIVES AS IMMUNOSTIMULANTS PFIZER INC. (US) 1994-05-18 EP disclosed
WO-1993003030-A1 QUINOLINE DERIVATIVES AS IMMUNOSTIMULANTS PFIZER INC. (US) 1993-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12528791-B2 Thyroid hormone receptor beta agonist compounds THRB, THRA, TSHR ESR1 1751/4885ESR2 248/4885ESRRB 149/4885
US-20220281849-A1 THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS THRB, THRA, TSHR ESR1 508/4885ESR2 135/4885ESRRB 92/4885
US-20260132121-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF RIPK1, RIPK2, RIPK4 ESR1 4074/4885ESR2 1948/4885ESRRB 2035/4885
US-12624018-B1 Inhibitors of RIPK2 and medical uses thereof RIPK2, RIPK1, RIPK4 ESR1 4773/4885ESR2 4201/4885ESRRB 4499/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.