SCHEMBL6163402

SCHEMBL6163402

CC(C)Cc1nn(C)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALPL P05186 2/20 0.45
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
OPRM1 P35372 10/20 0.38
HTT P42858 1/20 0.37
HSP90AA1 P07900 2/20 0.36
HSP90AB1 P08238 2/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166030 0.84 ALPL (0.40) ALPLALDH1A1KMT2ANPSR1HSD17B10
SCHEMBL6166123 0.82 ALPL (0.43) ALPLALDH1A1KMT2ANPSR1HSD17B10
SCHEMBL6162505 0.81 ALPL (0.67) ALPLALDH1A1KMT2ANPSR1HSD17B10
SCHEMBL6162256 0.78 OPRM1 (0.50) ALDH1A1KMT2ANPSR1HSD17B10OPRM1
SCHEMBL6166935 0.77 OPRM1 (0.39) ALPLKMT2AHSD17B10CRHBPCRHR2
SCHEMBL7479730 0.76 OPRM1 (0.54) ALDH1A1NPSR1OPRM1HSP90AA1HSP90AB1
SCHEMBL6769536 0.76 OPRM1 (0.51) ALDH1A1NPSR1OPRM1HSP90AA1HSP90AB1
SCHEMBL6167293 0.76 HTT (0.42) ALDH1A1OPRM1HTTLMNA
SCHEMBL6166168 0.74 OPRM1 (0.55) KMT2AHSD17B10OPRM1HTT
SCHEMBL6164703 0.74 OPRM1 (0.45) ALDH1A1KMT2ANPSR1OPRM1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed