SCHEMBL6165025

SCHEMBL6165025

O=C(CCc1cccnc1)NCCN1CCN(C(=O)N2c3ccccc3CCc3ccccc32)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
POLB P06746 1/20 0.43
C3AR1 Q16581 1/20 0.42
NAMPT P43490 2/20 0.42
OPRL1 P41146 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALOX15 P16050 1/20 0.41
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
CHRM1 P11229 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3080389 0.84 NAMPT (0.51) CYP1A2CYP3A4CYP2C9CYP2C19C3AR1
SCHEMBL21245369 0.79 HDAC8 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19NAMPT
Hydrochloric Acid SCHEMBL6164621 0.77 CYP3A4 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19POLB
SCHEMBL3077208 0.75 FNTA (0.47) CYP1A2CYP3A4CYP2C9CYP2C19C3AR1
SCHEMBL6482895 0.75 FNTA (0.47) CYP1A2CYP3A4CYP2C9CYP2C19C3AR1
SCHEMBL3458409 0.74 ALDH1A1 (0.63) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6271049 0.73 OPRL1 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19C3AR1
SCHEMBL7672874 0.72 CHRNA7 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL3458346 0.72 DRD2 (0.54) ALDH1A1DRD2DRD3
SCHEMBL83163 0.72 HTR1A (0.63) NAMPTHTR1AHTR7DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060163-B1 NEW PIPERAZINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES KLINGE CO CHEM PHARM FAB (DE) 2005-10-12 EP disclosed