SCHEMBL6165038

SCHEMBL6165038

CC(=O)N[C@@H](Cc1cccc(/C=N\N)c1)C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 4/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
PAM P19021 1/20 0.40
TACR1 P25103 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGB1 P05556 1/20 0.39
ITGAV P06756 1/20 0.39
ITGA2B P08514 1/20 0.39
ITGB5 P18084 1/20 0.39
PPARG P37231 1/20 0.38
GNPAT O15228 1/20 0.38
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
CAPN1 P07384 1/20 0.38
CTSB P07858 1/20 0.38
MMP1 P03956 1/20 0.37
FCER2 P06734 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6161741 0.92 HPGDS (0.40) HPGDSCTSSCTSKPAMTACR1
Trifluoroacetic Acid SCHEMBL6165425 0.78 CYP3A4 (0.45) HPGDSITGB3ITGB1ITGAVITGA2B
SCHEMBL15810862 0.76 CTSS (0.61) HPGDSCTSSCTSKPAMTACR1
SCHEMBL6248471 0.76 CTSS (0.61) HPGDSCTSSCTSKPAMTACR1
SCHEMBL15810860 0.76 CTSS (0.61) HPGDSCTSSCTSKPAMTACR1
SCHEMBL6165039 0.75 F10 (0.50) HPGDS
SCHEMBL6755037 0.74 POLB (0.42)
SCHEMBL6469894 0.72 TACR1 (0.62) TACR1FCER2
SCHEMBL18894273 0.72 ALOX15 (0.54) TACR1PPARG
SCHEMBL30493631 0.72 GNPAT (0.66) CTSSCTSKPAMGNPATMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP claimed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP claimed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO claimed