SCHEMBL6165784

SCHEMBL6165784

COC(=O)C(Cc1ccc(-c2nccs2)cc1)NC(=O)C(CSC(C)=O)Cc1ccccc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
DPP4 P27487 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
ABCC3 O15438 1/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
NR3C1 P04150 1/20 0.37
RARG P13631 1/20 0.37
CNR1 P21554 1/20 0.37
OPRK1 P41145 1/20 0.37
NR1H2 P55055 1/20 0.37
PPARA Q07869 1/20 0.37
NR1H3 Q13133 1/20 0.37
NR1I3 Q14994 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165788 1.00 KMT2A (0.42) KMT2ADPP4NPC1RAB9ACYP2C9
SCHEMBL6573642 0.90 CYP2C9 (0.47) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6575537 0.90 CYP2C9 (0.47) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6160498 0.86 PIN1 (0.41) NPC1RAB9ACYP2C9CYP2C19CYP1A2
SCHEMBL7324682 0.85 KMT2A (0.57) KMT2ACYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6161755 0.83 ABL1 (0.42) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6161753 0.83 ABL1 (0.42) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6160013 0.81 ALDH1A1 (0.44) RAB9ACYP2C9CYP2C19ALDH1A1THRB
SCHEMBL6161299 0.81 ALDH1A1 (0.44) RAB9ACYP2C9CYP2C19ALDH1A1THRB
SCHEMBL6160534 0.81 ALDH1A1 (0.44) RAB9ACYP2C9CYP2C19ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0877740-B1 THIOL DERIVATIVES WITH METALLOPEPTIDASE INHIBITORY ACTIVITY ZAMBON SPA (IT) 2005-03-30 EP disclosed