SCHEMBL6161753

SCHEMBL6161753

COC(=O)C(Cc1ccc(-c2nccs2)cc1)NC(=O)C(CSC(C)=O)Cc1cccc(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
POLB P06746 1/20 0.42
HDAC1 Q13547 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
ACE P12821 1/20 0.39
CTSD P07339 1/20 0.39
CTSA P10619 1/20 0.39
FFAR1 O14842 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ABCC3 O15438 1/20 0.39
NR1I2 O75469 1/20 0.39
ABCB11 O95342 1/20 0.39
NR3C1 P04150 1/20 0.39
RARG P13631 1/20 0.39
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161755 1.00 ABL1 (0.42) ABL1BCRPOLBHDAC1HDAC6
SCHEMBL6573642 0.91 CYP2C9 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6575537 0.91 CYP2C9 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6160498 0.90 PIN1 (0.41) HDAC1HDAC6CTSDFFAR1CYP1A2
SCHEMBL6165788 0.83 KMT2A (0.42) HDAC1HDAC6CYP1A2CYP3A4CYP2D6
SCHEMBL6165784 0.83 KMT2A (0.42) HDAC1HDAC6CYP1A2CYP3A4CYP2D6
SCHEMBL6161299 0.82 ALDH1A1 (0.44) CYP2C9CYP2C19
SCHEMBL6160013 0.82 ALDH1A1 (0.44) CYP2C9CYP2C19
SCHEMBL6160534 0.82 ALDH1A1 (0.44) CYP2C9CYP2C19
SCHEMBL6160968 0.82 ACE (0.52) ABL1BCRACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0877740-B1 THIOL DERIVATIVES WITH METALLOPEPTIDASE INHIBITORY ACTIVITY ZAMBON SPA (IT) 2005-03-30 EP disclosed