SCHEMBL6573642

SCHEMBL6573642

COC(=O)[C@H](Cc1ccc(-c2nccs2)cc1)NC(=O)[C@@H](CSC(C)=O)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
ABCC3 O15438 1/20 0.47
NR1I2 O75469 1/20 0.47
ABCB11 O95342 1/20 0.47
NR3C1 P04150 1/20 0.47
RARG P13631 1/20 0.47
CNR1 P21554 1/20 0.47
OPRK1 P41145 1/20 0.47
NR1H2 P55055 1/20 0.47
PPARA Q07869 1/20 0.47
NR1H3 Q13133 1/20 0.47
NR1I3 Q14994 1/20 0.47
ALDH1A1 P00352 1/20 0.45
THRB P10828 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MME P08473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575537 1.00 CYP2C9 (0.47) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6160534 0.91 ALDH1A1 (0.44) CYP2C9CYP2C19ALDH1A1THRBHSD17B10
SCHEMBL6161299 0.91 ALDH1A1 (0.44) CYP2C9CYP2C19ALDH1A1THRBHSD17B10
SCHEMBL6160013 0.91 ALDH1A1 (0.44) CYP2C9CYP2C19ALDH1A1THRBHSD17B10
SCHEMBL6161755 0.91 ABL1 (0.42) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6161753 0.91 ABL1 (0.42) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6160498 0.91 PIN1 (0.41) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6165784 0.90 KMT2A (0.42) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6165788 0.90 KMT2A (0.42) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6162656 0.86 MMP12 (0.43) CYP2C9CYP2C19ALDH1A1THRBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474405-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2004-11-10 EP disclosed
WO-2003068725-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-21 WO disclosed