SCHEMBL6167425

SCHEMBL6167425

N#Cc1ccc(-c2c(C(N)=O)cccc2-c2ccc(-c3ccccc3S(N)(=O)=O)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
F10 P00742 9/20 0.43
PARP1 P09874 3/20 0.43
PRSS1 P07477 2/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
PTGES2 Q9H7Z7 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
FABP1 P07148 1/20 0.40
BCAT2 O15382 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104689 0.90 ALOX5AP (0.42) F10PARP1PRSS1PRSS2PRSS3
SCHEMBL6165516 0.85 ALOX5AP (0.44) PARP1PARP2IRAK4
SCHEMBL6167423 0.78 F10 (0.62) F10PRSS1PRSS2PRSS3CA12
SCHEMBL8659145 0.78 CA1 (0.53) F10PTGES2CA12CA1CA2
SCHEMBL28045856 0.77 BCAT2 (0.65) PARP1PARP2IRAK4BCAT2
SCHEMBL6166620 0.76 ALOX5AP (0.44) F10PTGES2
SCHEMBL17593030 0.73 BCAT2 (0.49) PARP1PRSS1PRSS2PRSS3KEAP1
SCHEMBL2025737 0.73 BCAT2 (0.71) PARP1KEAP1NFE2L2BCAT2
SCHEMBL7112360 0.72 CA2 (0.56) F10PRSS1PRSS2PRSS3CA12
Hydrochloric Acid SCHEMBL27966297 0.71 BCAT2 (0.69) PARP1KEAP1NFE2L2BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP disclosed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP disclosed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO disclosed