SCHEMBL6167845

SCHEMBL6167845

Cc1ccc(S(=O)(=O)c2[nH]c3ccccc3c2/C=C/c2cccnc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
EGFR P00533 1/20 0.44
SRC P12931 1/20 0.44
NAMPT P43490 10/20 0.42
MAPT P10636 2/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
PADI4 Q9UM07 2/20 0.41
PLK4 O00444 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166809 0.77 EGFR (0.55) MEN1KMT2AALDH1A1TDP1EGFR
SCHEMBL6167611 0.75 NAMPT (0.46) MEN1KMT2AALDH1A1EGFRSRC
SCHEMBL18157727 0.74 CYP11B1 (0.53) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL5960508 0.73 EGFR (0.56) MEN1KMT2AALDH1A1TDP1EGFR
SCHEMBL20223300 0.72 CYP11B1 (0.58) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL20225455 0.70 CYP11B1 (0.51) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL4189420 0.70 EGFR (0.56) MEN1KMT2AALDH1A1TDP1EGFR
SCHEMBL9051693 0.69 EGFR (0.66) MEN1KMT2AALDH1A1TDP1EGFR
SCHEMBL6888612 0.69 CYP11B1 (0.70) MEN1KMT2AALDH1A1TDP1MAPT
SCHEMBL6166793 0.68 KDM4E (0.63) MEN1KMT2AALDH1A1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495016-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS MODULATORS OF P38 MAP KINASE Astex Technology Limited (GB) 2005-01-12 EP disclosed
WO-2003087087-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS MODULATORS OF P38 MAP KINASE ASTEX TECHNOLOGY LIMITED (GB) 2003-10-23 WO disclosed