SCHEMBL6168799

SCHEMBL6168799

COCCN1CCC(c2ccc(-c3ccccc3CO[C@@H](CC(C)C)C(=O)NCC#N)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSL P07711 8/20 0.41
CTSS P25774 8/20 0.41
CTSB P07858 7/20 0.41
CTSK P43235 6/20 0.41
PRCP P42785 2/20 0.41
SLC18A3 Q16572 1/20 0.39
HTR4 Q13639 1/20 0.38
CCR1 P32246 1/20 0.37
LRRK2 Q5S007 1/20 0.37
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5514860 0.90 CTSS (0.44) CTSLCTSSCTSBCTSKPRCP
SCHEMBL5509534 0.81 CTSL (0.44) CTSLCTSSCTSBCTSKPRCP
SCHEMBL5509530 0.81 CTSL (0.44) CTSLCTSSCTSBCTSKPRCP
SCHEMBL4700947 0.76 CTSL (0.66) CTSLCTSSCTSBCTSK
SCHEMBL6001121 0.76 CTSB (0.53) CTSLCTSSCTSBCTSK
SCHEMBL5515121 0.73 CTSS (0.40) CTSLCTSSCTSBCTSKDRD3
SCHEMBL5515117 0.73 CTSS (0.40) CTSLCTSSCTSBCTSKDRD3
SCHEMBL5515127 0.73 CTSS (0.40) CTSLCTSSCTSBCTSKDRD3
SCHEMBL4700791 0.73 CTSS (0.45) CTSLCTSSCTSBCTSK
SCHEMBL4700794 0.72 CTSS (0.62) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537074-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC. (CA) 2005-06-08 EP disclosed
WO-2004022526-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2004-03-18 WO disclosed