SCHEMBL6169928

SCHEMBL6169928

CCc1ccnc(C(=O)c2[nH]c3ccc(C(F)(F)F)cc3c2C(C)C(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.54
PTGS1 P23219 7/20 0.47
EGFR P00533 2/20 0.42
MRGPRX4 Q96LA9 2/20 0.38
GNRHR P30968 3/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
KIF11 P52732 1/20 0.36
CHUK O15111 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171474 0.89 PTGS2 (0.58) PTGS2PTGS1MEN1KMT2A
SCHEMBL6171485 0.87 PTGS2 (0.56) PTGS2PTGS1MEN1KMT2ATLR8
SCHEMBL6172077 0.87 PTGS2 (0.71) PTGS2PTGS1MEN1POLBKMT2A
SCHEMBL6171752 0.85 PTGS2 (0.49) PTGS2PTGS1MEN1KMT2A
SCHEMBL6169961 0.83 PTGS2 (0.76) PTGS2PTGS1EGFRMEN1KMT2A
SCHEMBL6174674 0.82 PTGS2 (0.68) PTGS2PTGS1EGFRMEN1KMT2A
SCHEMBL8113137 0.81 PTGS2 (0.55) PTGS2PTGS1EGFRMRGPRX4MEN1
SCHEMBL6174363 0.80 PTGS2 (0.49) PTGS2PTGS1MEN1KMT2A
SCHEMBL6170156 0.80 PTGS2 (0.50) PTGS2PTGS1KIF11
SCHEMBL7207232 0.79 PTGS2 (0.65) PTGS2PTGS1EGFRMRGPRX4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US disclosed