SCHEMBL6170699

SCHEMBL6170699

O=C(c1ccc(Cl)cc1)c1[nH]c2ccc(F)cc2c1C(C(=O)O)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 5/20 0.41
KDR P35968 2/20 0.41
AKR1C3 P42330 3/20 0.38
AKR1C2 P52895 3/20 0.38
PTGS2 P35354 3/20 0.38
MAPT P10636 2/20 0.38
PTGS1 P23219 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
ABCC4 O15439 1/20 0.38
C5 P01031 1/20 0.38
PDE4D Q08499 1/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CLK1 P49759 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171602 0.90 PTGS2 (0.46) MAP2PTGS2MAPTPTGS1KMT2A
SCHEMBL6171411 0.87 ALOX15 (0.47) MAP2MAPTKMT2AMEN1KDM4E
SCHEMBL6170687 0.85 MDM2 (0.43) PTGS2MAPTPTGS1KMT2AMEN1
SCHEMBL6172849 0.85 ALDH1A1 (0.42) MAP2PTGS2MAPTPTGS1KMT2A
SCHEMBL7202074 0.84 ALOX15 (0.42) AKR1C3AKR1C2PTGS2MAPTKMT2A
SCHEMBL6169060 0.82 GPR17 (0.44) PTGS2MAPTPTGS1KMT2AMEN1
SCHEMBL6169573 0.82 MEN1 (0.46) MAP2PTGS2KMT2AMEN1KDM4E
SCHEMBL6170210 0.79 MAP2 (0.46) MAP2PTGS2MAPTPTGS1KMT2A
SCHEMBL6169876 0.79 PTGS2 (0.46) PTGS2MAPTPTGS1KMT2AMEN1
SCHEMBL6168700 0.78 PTGS2 (0.58) AKR1C3AKR1C2PTGS2PTGS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP disclosed