SCHEMBL6170973

SCHEMBL6170973

Cc1nn(-c2ccccc2)nc1C(=O)N1CCCC1c1nnc(-c2ccncc2)o1.O=S(=O)(Cc1ccc(F)cc1F)N1CCCC1c1nnc(-c2cccnc2)o1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 18/20 0.42
HCRTR1 O43613 17/20 0.42
DPP4 P27487 1/20 0.35
SCD O00767 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364389 0.82 ALDH1A1 (0.44) DPP4SCD
SCHEMBL3366040 0.81 HCRTR1 (0.56) HCRTR2HCRTR1SCD
SCHEMBL6069077 0.73 ALDH1A1 (0.44) HCRTR2HCRTR1DPP4SCD
SCHEMBL3370704 0.71 HCRTR1 (0.63) HCRTR2HCRTR1
SCHEMBL3364395 0.71 ALDH1A1 (0.49)
SCHEMBL3369449 0.70 ALDH1A1 (0.46) DPP4
SCHEMBL3368142 0.69 CYP2C19 (0.44) HCRTR2HCRTR1DPP4
SCHEMBL3367004 0.67 CYP2C19 (0.41) HCRTR2HCRTR1
SCHEMBL3370780 0.67 CYP2C19 (0.41) HCRTR2HCRTR1
SCHEMBL3366667 0.67 KDM4E (0.43) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-A1 2-PYRROLIDIN-2-YL- 1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS Grünenthal GmbH (DE) 2005-05-25 EP disclosed
WO-2004024725-A1 2-PYRROLIDIN-2-YL-[1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS Grünenthal GmbH (DE) 2004-03-25 WO disclosed