SCHEMBL6172425

SCHEMBL6172425

CCN(C(=O)Oc1ccccc1)c1ccc(-n2nc(C)c(-c3ccccc3)c2C)nc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OXTR P30559 3/20 0.39
MAPT P10636 7/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
RAB9A P51151 2/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
TP53 P04637 2/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6172823 0.86 RAB9A (0.47) OXTRMAPTLMNANPSR1RAB9A
SCHEMBL6172817 0.82 MAPT (0.43) MAPTKMT2ALMNANPSR1RAB9A
SCHEMBL6097690 0.74 MEN1 (0.53) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL6096779 0.70 NPC1 (0.40) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL4089380 0.69 ALDH1A1 (0.61) MAPTMEN1KMT2ANPSR1RAB9A
SCHEMBL6096848 0.66 KDM4E (0.42) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL3683672 0.65 ALDH1A1 (0.50) MAPTNPSR1RAB9AKDM4EALDH1A1
SCHEMBL6100494 0.65 CHRNB2 (0.43) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL9267264 0.64 ALDH1A1 (0.56) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL13341592 0.63 KMT2A (0.41) MAPTMEN1KMT2ARAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495005-A1 PYRAZOLE COMPOUNDS AS ANTI-INFLAMMATORY AND ANALGESIC AGENTS Pfizer Japan Inc. (JP) 2005-01-12 EP disclosed
WO-2003087061-A1 PYRAZOLE COMPOUNDS AS ANTI-INFLAMMATORY AND ANALGESIC AGENTS PFIZER JAPAN INC. (JP) 2003-10-23 WO disclosed