SCHEMBL6176017

SCHEMBL6176017

Cc1ccc2c(c1)N(CC(=O)C(C)(C)C)C(=O)C(N)CN2c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CCKBR P32239 2/20 0.36
THRB P10828 1/20 0.36
AADAT Q8N5Z0 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6176423 0.89 ALDH1A1 (0.48) CCKARALDH1A1CCKBRTHRB
SCHEMBL1394353 0.89 ALDH1A1 (0.48) CCKARALDH1A1CCKBRTHRB
SCHEMBL7959523 0.87 TSHR (0.39) ALDH1A1CCKBRAADAT
Oxalic Acid SCHEMBL6825177 0.86 ALDH1A1 (0.46) CCKARALDH1A1CCKBRTHRB
Oxalic Acid SCHEMBL6825172 0.86 ALDH1A1 (0.46) CCKARALDH1A1CCKBRTHRB
SCHEMBL6176919 0.81 CCKBR (0.42) CCKARCCKBR
SCHEMBL6177886 0.80 MMP2 (0.50) CCKBR
SCHEMBL6179020 0.80 MMP2 (0.50) CCKBR
SCHEMBL6181517 0.78 CCKBR (0.43) CCKARALDH1A1CCKBRAADAT
SCHEMBL6175868 0.76 CCKBR (0.58) CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945445-B9 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2005-12-28 EP disclosed
EP-0945445-B1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2003-09-03 EP disclosed
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed
EP-0945445-A1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed