SCHEMBL6178527

SCHEMBL6178527

CCCC(C)(NC(=O)Cc1ccc(NC(=O)Nc2ccccc2C)cc1)C(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.51
ITGA4 P13612 14/20 0.51
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
HPGD P15428 1/20 0.47
RORC P51449 1/20 0.44
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
GHSR Q92847 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180128 0.87 ITGB1 (0.56) ITGB1ITGA4RAB9ANPC1HPGD
SCHEMBL6178535 0.77 ITGB1 (0.55) ITGB1ITGA4
SCHEMBL6177419 0.74 ITGB1 (0.63) ITGB1ITGA4
SCHEMBL3485567 0.73 ITGB1 (0.67) ITGB1ITGA4RAB9ANPC1HPGD
SCHEMBL29612679 0.73 ITGB1 (0.67) ITGB1ITGA4RAB9ANPC1HPGD
SCHEMBL8236504 0.71 ITGB1 (0.56) ITGB1ITGA4RAB9ANPC1HPGD
SCHEMBL18472821 0.71 ITGB1 (0.58) ITGB1ITGA4RAB9ANPC1HPGD
SCHEMBL8231040 0.71 ITGB1 (0.61) ITGB1ITGA4RAB9ANPC1HPGD
SCHEMBL14561170 0.70 RAB9A (0.67) ITGB1ITGA4RAB9ANPC1MAPT
SCHEMBL17477398 0.70 POLB (0.48) HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091943-B1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PROD INC (US) 2005-11-30 EP disclosed
US-6355662-B1 PEPTIDE AND NONPEPTIDES AUTOIMMUNE DISEASES, ANTIINFLAMMATORY AGENTS PFIZER INC 2002-03-12 US disclosed
US-6306887-B1 AROMATIC UREAS, CARBAMATES AND TRIAMINONITRILES AND HETEROCYCLIC COMPOUNDS PFIZER INC 2001-10-23 US disclosed
EP-1091943-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES Pfizer Products Inc. (US) 2001-04-18 EP disclosed
WO-2000000477-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PRODUCTS INC. (US) 2000-01-06 WO disclosed