SCHEMBL6179501

SCHEMBL6179501

CN(C(=O)CN1C(=O)C(N)CN(c2ccccc2)c2ccccc21)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 5/20 0.45
CCKBR P32239 5/20 0.45
POLB P06746 1/20 0.41
DRD4 P21917 1/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TSHR P16473 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180449 0.86 CCKAR (0.44) CCKARCCKBRPOLBDRD4NPC1
SCHEMBL6181562 0.81 POLB (0.48) CCKARCCKBRPOLBDRD4NPC1
SCHEMBL6176423 0.81 ALDH1A1 (0.48) CCKARCCKBRPOLBALDH1A1
SCHEMBL1394353 0.81 ALDH1A1 (0.48) CCKARCCKBRPOLBALDH1A1
Oxalic Acid SCHEMBL6825172 0.78 ALDH1A1 (0.46) CCKARCCKBRPOLBALDH1A1
SCHEMBL6177759 0.78 CCKBR (0.43) CCKARCCKBRNPC1ALDH1A1
SCHEMBL6178095 0.78 MAPT (0.42) CCKBR
SCHEMBL6179137 0.78 CYP3A4 (0.40) CCKBRNPC1RAB9ATSHRALDH1A1
Oxalic Acid SCHEMBL6825177 0.78 ALDH1A1 (0.46) CCKARCCKBRPOLBALDH1A1
SCHEMBL6180398 0.78 CCKAR (0.44) CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945445-B9 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2005-12-28 EP disclosed
EP-0945445-B1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2003-09-03 EP disclosed
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed
EP-0945445-A1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed