SCHEMBL6180572

SCHEMBL6180572

COCCC(=O)Nc1ccc(N2CC3CCC2CC3)c(OC(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.43
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
F2R P25116 1/20 0.40
EPHX2 P34913 5/20 0.39
S1PR2 O95136 1/20 0.38
AAK1 Q2M2I8 1/20 0.37
BACE1 P56817 1/20 0.36
GSTO1 P78417 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1379964 0.83 CYP2D6 (0.47) MCHR1NPSR1KDM4EAAK1
SCHEMBL4479717 0.78 F10 (0.55)
SCHEMBL4033308 0.78 F10 (0.55)
SCHEMBL4033674 0.66 SMN1; SMN2 (0.35)
SCHEMBL20679611 0.62 GSTO1 (0.63) NPSR1KDM4EEPHX2GSTO1
SCHEMBL30675599 0.62 GSTO1 (0.63) NPSR1KDM4EEPHX2GSTO1
SCHEMBL6181130 0.61 F10 (0.66) GSTO1
SCHEMBL1377310 0.61 F10 (0.61) KDM4EBACE2
SCHEMBL5873685 0.61 MCHR1 (0.59) MCHR1EPHX2
SCHEMBL7873626 0.61 NPSR1 (0.57) MCHR1NPSR1KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562939-A1 CARBOXAMIDES MERCK PATENT GmbH (DE) 2005-08-17 EP disclosed
WO-2004046138-A1 CARBOXAMIDES MERCK PATENT GMBH (DE) 2004-06-03 WO disclosed