SCHEMBL6180637

SCHEMBL6180637

Cc1ccc2c(c1)CC(C1=CNC(=S)[N]1)C2

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801994 0.82 SLC6A4 (0.38)
SCHEMBL5802511 0.81 ADRA1A (0.39)
SCHEMBL5798860 0.72 PLAU (0.39)
SCHEMBL5802586 0.69 ADRA1A (0.32)
SCHEMBL1340369 0.66 UBE2N (0.36) ACHE
SCHEMBL13241438 0.64 ACHE (0.44) ACHEPDE3BPDE3A
SCHEMBL13241439 0.64 ACHE (0.44) ACHEPDE3BPDE3A
SCHEMBL18826051 0.64 ADRA2A (0.46)
SCHEMBL80428 0.64 ACHE (0.47) ACHE
SCHEMBL31236154 0.64 ACHE (0.47) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507767-A1 4-SUBSTITUTED IMIDAZOLE-2-THIONES AND IMIDAZOL-2-ONES AS AGONISTS OF THE ALPHA-2B AND ALPHA-2C ADRENERGIC RECEPTORS Allergan, Inc. (US) 2005-02-23 EP disclosed
WO-2003099795-A1 4-SUBSTITUTED IMIDAZOLE-2-THIONES AND IMIDAZOL-2-ONES AS AGONISTS OF THE ALPHA-2B AND ALPHA-2C ADRENERGIC RECEPTORS ALLERGAN, INC. (US) 2003-12-04 WO disclosed