SCHEMBL6181701

SCHEMBL6181701

O=C(NC1CN(C(=O)C2CCCCC2)c2ccccc2N(c2ccccc2)C1=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
EPHX1 P07099 1/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.41
CASP3 P42574 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NAAA Q02083 3/20 0.40
ASAH1 Q13510 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSK P43235 1/20 0.40
PREP P48147 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178886 0.83 CTSK (0.43) GAANAAACTSLCTSBCTSK
SCHEMBL6178514 0.82 GAA (0.47) ALDH1A1EPHX1GAATSHRMEN1
SCHEMBL6181018 0.81 CCKBR (0.43) CASP3
SCHEMBL7962877 0.76 NAAA (0.54) NAAAASAH1CTSL
SCHEMBL10937277 0.74 NAAA (0.55) ALDH1A1EPHX1GAATSHRNAAA
SCHEMBL9740624 0.74 NAAA (0.55) ALDH1A1EPHX1GAATSHRNAAA
SCHEMBL8342642 0.74 GAA (0.63) ALDH1A1GAAMEN1KMT2ANAAA
SCHEMBL10945585 0.73 NAAA (0.50) ALDH1A1EPHX1GAATSHRCASP3
SCHEMBL10832788 0.73 PREP (0.52) ALDH1A1GAATSHRNAAACTSL
SCHEMBL10832792 0.73 PREP (0.52) ALDH1A1GAATSHRNAAACTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945445-B9 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2005-12-28 EP disclosed
EP-0945445-B1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2003-09-03 EP disclosed
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed
EP-0945445-A1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed