SCHEMBL6182589

SCHEMBL6182589

COC(=O)c1cc(-c2ccncc2)ncc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 1/20 0.52
AXL P30530 1/20 0.49
CASP1 P29466 4/20 0.47
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
HPGDS O60760 1/20 0.43
AAK1 Q2M2I8 2/20 0.43
NR4A2 P43354 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PPARG P37231 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6181603 0.81 DHODH (0.47) CASP1ALDH1A1GAAPPARGMAPT
SCHEMBL16635187 0.77 MAPT (0.42) CASP1ALDH1A1KDM4EGAAKMT2A
SCHEMBL17987105 0.77 CNR1 (0.35) AXLALDH1A1KDM4EGAAMEN1
SCHEMBL25148607 0.75 LDHA (0.54) AXLALDH1A1KDM4EGAANR4A2
SCHEMBL11379519 0.75 AXL (0.60) CYP46A1AXLCASP1ALDH1A1KDM4E
SCHEMBL30364708 0.75 LDHA (0.54) AXLALDH1A1KDM4EGAANR4A2
SCHEMBL30217866 0.75 KDM4E (0.47) ALDH1A1KDM4EGLAGAAMEN1
SCHEMBL31598658 0.75 ALDH1A1 (0.64) CYP46A1CASP1ALDH1A1KDM4EGLA
SCHEMBL236107 0.75 KDM4E (0.47) ALDH1A1KDM4EGLAGAAMEN1
SCHEMBL949750 0.75 ALDH1A1 (0.64) CYP46A1CASP1ALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501805-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2005-02-02 EP disclosed
WO-2003095430-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2003-11-20 WO disclosed