SCHEMBL6182737

SCHEMBL6182737

Cc1ccc(C(Cl)C=O)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
POLB P06746 2/20 0.42
AKR1C3 P42330 2/20 0.41
AKR1C2 P52895 2/20 0.41
TP53 P04637 1/20 0.40
LMNA P02545 5/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
HTT P42858 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ERN1 O75460 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
DAO P14920 1/20 0.33
GPR139 Q6DWJ6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247899 0.82 CES2 (0.42) ALDH1A1AKR1C3AKR1C2
SCHEMBL20495193 0.82 CES2 (0.42) ALDH1A1AKR1C3AKR1C2
SCHEMBL18942465 0.79 AKR1C3 (0.45) ALDH1A1POLBAKR1C3AKR1C2TP53
SCHEMBL19555328 0.79 PSEN1 (0.36) ALDH1A1GPR139
SCHEMBL17165350 0.79 PSEN1 (0.36) ALDH1A1GPR139
SCHEMBL5702253 0.79 SHBG (0.46) LMNAERN1
SCHEMBL12492053 0.78 KDM1A (0.33)
SCHEMBL27605593 0.77 LMNA (0.40) ALDH1A1POLBAKR1C3AKR1C2TP53
SCHEMBL8282398 0.74 AKR1C3 (0.41) ALDH1A1POLBAKR1C3AKR1C2TP53
SCHEMBL22031605 0.73 OPRM1 (0.39) ALDH1A1POLBAKR1C3AKR1C2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507530-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-02-23 EP disclosed
WO-2003097048-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-27 WO disclosed