SCHEMBL6182783

SCHEMBL6182783

CCOC(=O)c1ccnc(C#N)c1C#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.48
ALDH1A1 P00352 4/20 0.48
HSD17B10 Q99714 4/20 0.48
MAPT P10636 3/20 0.48
NUDT1 P36639 1/20 0.48
GLA P06280 1/20 0.48
ATM Q13315 1/20 0.48
KMT2A Q03164 1/20 0.47
ALOX15 P16050 2/20 0.47
GAA P10253 2/20 0.47
TP53 P04637 1/20 0.47
APOBEC3G Q9HC16 1/20 0.47
L3MBTL1 Q9Y468 6/20 0.45
TSHR P16473 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TDP1 Q9NUW8 1/20 0.43
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
ELANE P08246 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25370390 0.85 NUDT1 (0.48) KDM4EALDH1A1HSD17B10MAPTNUDT1
SCHEMBL2800784 0.81 TSHR (0.54) KDM4EALDH1A1HSD17B10KMT2AGAA
SCHEMBL9236279 0.78 TSHR (0.63) KDM4EALDH1A1HSD17B10MAPTGLA
SCHEMBL25373071 0.77 L3MBTL1 (0.47) KDM4EALDH1A1HSD17B10KMT2AALOX15
SCHEMBL10568384 0.73 NLRP3 (0.48) ALDH1A1ATMTSHRSMN1; SMN2POLB
SCHEMBL7870053 0.73 TSHR (0.56) KDM4EALDH1A1HSD17B10MAPTGLA
SCHEMBL29151319 0.73 CA12 (0.51) KDM4EALDH1A1HSD17B10MAPTGLA
SCHEMBL109089 0.72 TSHR (0.54) KDM4EALDH1A1HSD17B10MAPTGLA
SCHEMBL9476717 0.72 ALDH1A1 (0.51) KDM4EALDH1A1HSD17B10MAPTGLA
SCHEMBL25372176 0.71 NLRP3 (0.36) KDM4EALDH1A1HSD17B10MAPTNUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501805-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2005-02-02 EP disclosed
WO-2003095430-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2003-11-20 WO disclosed