SCHEMBL6184565

SCHEMBL6184565

CN(C(=O)Cc1cccc(Br)c1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.48
ERBB2 P04626 1/20 0.48
POLQ O75417 4/20 0.47
PTGES O14684 1/20 0.46
TAAR1 Q96RJ0 1/20 0.45
RIPK1 Q13546 1/20 0.45
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
NLRP3 Q96P20 1/20 0.44
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
KMT2A Q03164 1/20 0.43
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8263373 0.84 ALDH1A1 (0.58) POLQALDH1A1LMNAROCK2ROCK1
SCHEMBL20349603 0.83 ALDH1A1 (0.52) POLQALDH1A1LMNANLRP3ROCK2
SCHEMBL5240155 0.82 TAAR1 (0.51) EGFRERBB2PTGESTAAR1RIPK1
SCHEMBL11630604 0.82 OPRK1 (0.52) POLQALDH1A1LMNANLRP3ROCK2
SCHEMBL20346359 0.82 POLQ (0.47) POLQALDH1A1LMNANLRP3ROCK2
SCHEMBL5461014 0.77 SIGMAR1 (0.56) ALDH1A1LMNAKDM4E
SCHEMBL1515805 0.77 TAAR1 (0.46) EGFRERBB2PTGESTAAR1RIPK1
SCHEMBL15676809 0.77 SIGMAR1 (0.56) ALDH1A1LMNAKMT2A
SCHEMBL4247854 0.76 RAB9A (0.50) EGFRERBB2PTGESTAAR1RIPK1
SCHEMBL11630235 0.76 ALDH1A1 (0.48) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6927228-B2 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-09 US disclosed
EP-1309575-B1 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS GALDERMA RES & DEV (FR) 2005-06-08 EP disclosed
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors PPARG, PPARA, PPARD EGFR 1435/4885ERBB2 704/4885POLQ 1557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.