SCHEMBL6184923

SCHEMBL6184923

NC(=O)Cc1ccccc1-c1ccc(Cl)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.64
FGFR1 P11362 1/20 0.46
SRC P12931 1/20 0.46
FGFR2 P21802 1/20 0.46
FGFR4 P22455 1/20 0.46
FGFR3 P22607 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
FFAR4 Q5NUL3 2/20 0.46
FFAR1 O14842 1/20 0.46
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
PTGS2 P35354 2/20 0.45
PTGS1 P23219 1/20 0.45
SUCNR1 Q9BXA5 2/20 0.43
KMT2A Q03164 1/20 0.42
GCG P01275 1/20 0.41
ACLY P53396 1/20 0.41
F10 P00742 2/20 0.40
DPP4 P27487 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7598404 0.88 CYP2C19 (0.54) CYP2C19FGFR1SRCFGFR2FGFR4
SCHEMBL1547038 0.85 KMT2A (0.56) CYP2C19PTGDR2FFAR4FFAR1KMT2A
SCHEMBL2391279 0.85 CYP2C19 (0.48) CYP2C19KMT2AACLY
SCHEMBL3540535 0.84 SUCNR1 (0.56) CYP2C19PTGDR2FFAR4FFAR1SLC6A4
Hydrochloric Acid SCHEMBL27396597 0.84 KMT2A (0.55) CYP2C19PTGDR2FFAR4FFAR1KMT2A
SCHEMBL7311559 0.84 BCAT2 (0.50) CYP2C19PTGS1KMT2AACLYDPP4
SCHEMBL2391344 0.83 FFAR1 (0.46) CYP2C19FFAR4FFAR1SLC6A3KMT2A
SCHEMBL2392196 0.83 PTGDR2 (0.46) CYP2C19PTGDR2FFAR4FFAR1SLC6A4
SCHEMBL2395091 0.83 CYP2C19 (0.49) CYP2C19FFAR4FFAR1ACLYNPC1
SCHEMBL2393760 0.82 CHRM1 (0.56) CYP2C19ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
EP-2374790-A1 BIPHENYLACETAMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2011-10-12 EP disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed
EP-1567502-A1 SUBSTITUTED DIHYDROPHENANTHRIDINESUL FONAMIDES Wyeth (US) 2005-08-31 EP disclosed
WO-2004050631-A1 SUBSTITUTED DIHYDROPHENANTHRIDINESUL FONAMIDES WYETH (US) 2004-06-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE HRH3, KCNH3, BRPF3 CYP2C19 240/4885FGFR1 294/4885SRC 2996/4885
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE HRH3, KCNH3, BRPF3 CYP2C19 240/4885FGFR1 294/4885SRC 2996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.