SCHEMBL6189630

SCHEMBL6189630

CC/C(=C(/C)C(=O)O)c1ccccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
ERCC5 P28715 2/20 0.50
FEN1 P39748 2/20 0.50
TP53 P04637 1/20 0.49
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
HPGD P15428 2/20 0.45
POLB P06746 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ESR1 P03372 1/20 0.40
TSHR P16473 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28419366 0.82 CLCN2 (0.41) ALDH1A1ERCC5FEN1CES2CES1
SCHEMBL30931566 0.79 ALDH1A1 (0.57) ALDH1A1ERCC5FEN1TP53CES2
SCHEMBL4624841 0.78 NR4A1 (0.53) ALDH1A1TP53HPGDPOLBSMN1; SMN2
SCHEMBL7174103 0.77 CES2 (0.50) CES2CES1SMN1; SMN2ESR1
SCHEMBL349595 0.77 CES2 (0.50) CES2CES1SMN1; SMN2ESR1
SCHEMBL5279624 0.77 CES2 (0.50) CES2CES1SMN1; SMN2ESR1
SCHEMBL2837238 0.75 ERCC5 (0.58) ALDH1A1ERCC5FEN1TP53CES2
Water SCHEMBL7994046 0.73 ERCC5 (0.56) ALDH1A1ERCC5FEN1TP53CES2
Hydrochloric Acid SCHEMBL30461901 0.73 ERCC5 (0.56) ALDH1A1ERCC5FEN1TP53CES2
Acetic Acid SCHEMBL9331813 0.72 ALDH1A1 (0.86) ALDH1A1ERCC5FEN1TP53CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041980-B1 ACYL GUANIDINE SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL MYERS SQUIBB CO (US) 2005-02-23 EP disclosed
EP-1041980-A4 ACYL GUANIDINE SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL MYERS SQUIBB CO (US) 2002-03-20 EP disclosed
EP-1041980-A1 ACYL GUANIDINE SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2000-10-11 EP disclosed
US-6011059-A PREVENTING OR TREATING ANGINA PECTORIS, CARDIAC DYSFUNCTION, MYOCARDIAL NECROSIS, AND ARRHYTHMIA EMPLOYING THE ABOVE ACYL GUANIDINES. BRISTOL-MYERS SQUIBB COMPANY (US) 2000-01-04 US disclosed
WO-1999033460-A1 ACYL GUANIDINE SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 1999-07-08 WO disclosed