SCHEMBL6192513

SCHEMBL6192513

COc1ccc(CC(=O)N2CCN(S(=O)(=O)c3cccc4cccnc34)C(C(=O)NCC(c3ccccc3)c3ccccc3)C2)cc1.O=C(NCC(c1ccccc1)c1ccccc1)C1CN(C(=O)CCN2CCCCC2)CCN1S(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
MAPK1 P28482 3/20 0.46
GAA P10253 3/20 0.46
LMNA P02545 2/20 0.45
HSP90AA1 P07900 1/20 0.45
HTT P42858 1/20 0.43
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 4/20 0.41
TSHR P16473 2/20 0.41
POLB P06746 2/20 0.41
GFER P55789 1/20 0.41
MMP1 P03956 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036850 0.93 ALDH1A1 (0.52) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL4035069 0.91 GAA (0.53) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL4032496 0.88 ALDH1A1 (0.51) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL4035404 0.84 GAA (0.55) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL4038343 0.82 GAA (0.57) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL4036852 0.80 MMP1 (0.50) ALDH1A1SMN1; SMN2GAALMNAHTT
SCHEMBL4034935 0.79 ALDH1A1 (0.51) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL4035075 0.77 CHRM1 (0.40) ALDH1A1HPGDSMN1; SMN2GAALMNA
SCHEMBL4033651 0.77 GAA (0.56) ALDH1A1HPGDSMN1; SMN2MAPK1GAA
SCHEMBL1384878 0.77 ALDH1A1 (0.55) ALDH1A1HPGDSMN1; SMN2MAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2005-11-09 EP claimed
WO-2004071390-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-08-26 WO claimed