SCHEMBL6198529

SCHEMBL6198529

O=[N+]([O-])c1ccc(COCCOCc2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2C19 P33261 1/20 0.57
RAB9A P51151 2/20 0.54
NPC1 O15118 1/20 0.54
ALDH1A1 P00352 3/20 0.52
LMNA P02545 1/20 0.52
AKR1C3 P42330 1/20 0.51
PTPRF P10586 1/20 0.51
PTPN2 P17706 1/20 0.51
PTPN1 P18031 1/20 0.51
PTPN11 Q06124 1/20 0.51
HTT P42858 1/20 0.51
MAPT P10636 3/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19621588 0.93 IDO1 (0.61) IDO1CYP1A2CYP2C19RAB9ANPC1
SCHEMBL11441117 0.93 IDO1 (0.61) IDO1CYP1A2CYP2C19RAB9ANPC1
SCHEMBL7931694 0.92 IDO1 (0.53) IDO1CYP1A2CYP2C19RAB9ANPC1
SCHEMBL27712803 0.91 TSHR (0.60) IDO1CYP1A2CYP2C19RAB9ANPC1
SCHEMBL4758638 0.89 DRD2 (0.57) CYP2C19ALDH1A1LMNAHTTMAPT
SCHEMBL1164057 0.86 TDP1 (0.59) IDO1CYP1A2CYP2C19RAB9ANPC1
Ether SCHEMBL11441077 0.85 IDO1 (0.53) IDO1CYP1A2CYP2C19RAB9ANPC1
SCHEMBL37463 0.85 IDO1 (0.70) IDO1CYP1A2CYP2C19RAB9AALDH1A1
P-Nitrophenol SCHEMBL9638804 0.84 NPC1 (0.56) IDO1CYP1A2CYP2C19RAB9ANPC1
SCHEMBL12478072 0.84 IDO1 (0.56) IDO1RAB9AALDH1A1LMNAAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042295-B1 4-HYDROXYQUINOLINE-3-CARBOXAMIDES AND HYDRAZIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN CO LLC (US) 2005-09-07 EP disclosed
EP-1042295-A1 4-HYDROXYQUINOLINE-3-CARBOXAMIDES AND HYDRAZIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-10-11 EP disclosed
US-6093732-A PREVENT HERPESVIRAL INFECTIONS, PARTICULARLY, HUMAN CYTOMEGALOVIRAL INFECTION PHARMACIA & UPJOHN COMPANY (US) 2000-07-25 US disclosed
WO-1999032450-A1 4-HYDROXYQUINOLINE-3-CARBOXAMIDES AND HYDRAZIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-01 WO disclosed