SCHEMBL6199517

SCHEMBL6199517

COc1ccc(S(=O)(=O)N[C@](Cc2ccccc2)(NC(=O)O)[C@@H](C)O)cc1CC(C)(C)CCN

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
PKM P14618 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
F2 P00734 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CTSD P07339 2/20 0.35
MMP1 P03956 1/20 0.35
MMP9 P14780 1/20 0.35
MMP13 P45452 1/20 0.35
HSD17B10 Q99714 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5770229 0.86 HTR6 (0.34) HTR6SMN1; SMN2PKMCYP3A4CYP2C19
SCHEMBL7569774 0.84 MEN1 (0.32) HTR6SMN1; SMN2PKMCYP3A4CYP2C19
SCHEMBL1602534 0.82 ABCB1 (0.46) CYP3A4CTSDALDH1A1MAPTKMT2A
SCHEMBL5772049 0.82 ABCB1 (0.46) CYP3A4CTSDALDH1A1MAPTKMT2A
SCHEMBL1600751 0.82 ABCB1 (0.46) CYP3A4CTSDALDH1A1MAPTKMT2A
SCHEMBL1601307 0.79 ABCB1 (0.45) KMT2A
SCHEMBL1602713 0.79 ABCB1 (0.45) KMT2A
SCHEMBL1603130 0.72 ABCB1 (0.42) KMT2A
SCHEMBL1600573 0.72 ABCB1 (0.41) KMT2A
SCHEMBL5771962 0.69 MMP1 (0.34) HTR6MMP1MMP9MMP13ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159278-B1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMA (US) 2005-11-30 EP disclosed