SCHEMBL5770229

SCHEMBL5770229

COc1ccc(S(=O)(=O)N[C@](Cc2ccccc2)(NC(=O)Oc2ccoc2)[C@@H](C)O)cc1CC(C)(C)CCN

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.34
CASP1 P29466 1/20 0.32
CASP3 P42574 1/20 0.32
CASP7 P55210 1/20 0.32
CASP8 Q14790 1/20 0.32
MGAT2 Q10469 1/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
ITGAV P06756 2/20 0.32
ALDH1A1 P00352 2/20 0.32
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
HDAC1 Q13547 1/20 0.31
TNF P01375 1/20 0.31
NOD2 Q9HC29 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6199517 0.86 HTR6 (0.38) HTR6MMP1MMP9MMP13ALDH1A1
SCHEMBL7569774 0.85 MEN1 (0.32) HTR6ALDH1A1PKMSMN1; SMN2KMT2A
SCHEMBL5771962 0.84 MMP1 (0.34) HTR6CASP1CASP3CASP7CASP8
SCHEMBL5771240 0.81 MMP1 (0.33) HTR6CASP1CASP3CASP7CASP8
SCHEMBL1602534 0.78 ABCB1 (0.46) ALDH1A1KMT2ACYP3A4
SCHEMBL5772049 0.78 ABCB1 (0.46) ALDH1A1KMT2ACYP3A4
SCHEMBL1600751 0.78 ABCB1 (0.46) ALDH1A1KMT2ACYP3A4
SCHEMBL1602713 0.75 ABCB1 (0.45) KMT2A
SCHEMBL1601307 0.75 ABCB1 (0.45) KMT2A
SCHEMBL5771487 0.74 KMT2A (0.33) CASP1CASP3CASP7CASP8MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637518-A2 Inhibitors of aspartyl protease Vertex Pharmaceuticals Incorporated (US) 2006-03-22 EP disclosed