SCHEMBL5771962

SCHEMBL5771962

COc1ccc(S(=O)(=O)[C@@](C)(O)[C@](N)(Cc2ccccc2)NC(=O)Oc2ccoc2)cc1CC(C)(C)CCN

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 3/20 0.34
MMP13 P45452 3/20 0.34
MMP9 P14780 2/20 0.34
KMT2A Q03164 1/20 0.33
HTR6 P50406 1/20 0.33
TAS2R14 Q9NYV8 2/20 0.32
ALDH1A1 P00352 2/20 0.31
CASP1 P29466 1/20 0.30
CASP3 P42574 1/20 0.30
CASP7 P55210 1/20 0.30
CASP8 Q14790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5771240 0.96 MMP1 (0.33) MMP1MMP13MMP9KMT2AHTR6
SCHEMBL5770229 0.84 HTR6 (0.34) MMP1MMP13MMP9KMT2AHTR6
SCHEMBL5771968 0.81 MMP1 (0.44) MMP1MMP13MMP9ALDH1A1
SCHEMBL5771246 0.78 MMP1 (0.42) MMP1MMP13MMP9ALDH1A1
SCHEMBL5773477 0.77 ABCB1 (0.43) KMT2A
SCHEMBL5773719 0.77 ABCB1 (0.43) KMT2A
SCHEMBL5771712 0.74 ABCB1 (0.42)
SCHEMBL5772320 0.74 ABCB1 (0.42)
SCHEMBL5771487 0.71 KMT2A (0.33) MMP9KMT2ATAS2R14CASP1CASP3
SCHEMBL7569774 0.70 MEN1 (0.32) KMT2AHTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637518-A2 Inhibitors of aspartyl protease Vertex Pharmaceuticals Incorporated (US) 2006-03-22 EP disclosed