SCHEMBL6201346

SCHEMBL6201346

CCOC(=O)C(c1ccccc1)c1cn[nH]c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.48
LMNA P02545 2/20 0.48
CYP2D6 P10635 1/20 0.48
CYP3A4 P08684 3/20 0.47
GABRA1 P14867 2/20 0.47
GABRB2 P47870 2/20 0.47
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ABCB11 O95342 1/20 0.47
GABRA2 P47869 1/20 0.47
CHRM1 P11229 4/20 0.47
CHRM3 P20309 4/20 0.47
CHRM2 P08172 3/20 0.47
CHRM4 P08173 3/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9327799 0.85 KMT2A (0.50) CYP1A2LMNACYP2D6CHRM1CHRM3
SCHEMBL2310025 0.84 LMNA (0.62) CYP1A2LMNACYP2D6CYP3A4CHRM1
SCHEMBL1560439 0.81 AKT2 (0.41) LMNACYP2D6L3MBTL1
SCHEMBL6055220 0.78 MEN1 (0.43) CYP1A2CYP2D6ALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL4534323 0.78 CYP1A2 (0.53) CYP1A2LMNACYP2D6CYP3A4GABRA1
SCHEMBL9326757 0.78 MEN1 (0.43) CYP1A2CYP2D6ALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL5084136 0.78 LMNA (0.55) CYP1A2LMNACYP2D6CYP3A4CHRM1
SCHEMBL30350798 0.76 NOS2 (0.41) CYP1A2LMNACYP3A4GABRA1GABRB2
SCHEMBL27965729 0.76 LMNA (0.54) CYP1A2LMNACYP2D6CYP3A4CHRM1
SCHEMBL29299737 0.75 LMNA (0.53) CYP1A2LMNACYP2D6CYP3A4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562937-A2 N-SUBSTITUTED PIPERIDINE DERIVATIVES AS SEROTONIN RECEPTOR AGENTS Acadia Pharmaceuticals Inc. (US) 2005-08-17 EP disclosed
WO-2004000808-A2 N-SUBSTITUTED PIPERIDINE DERIVATIVES AS SEROTONIN RECEPTOR AGENTS ACADIA PHARMACEUTICALS INC. (US) 2003-12-31 WO disclosed