SCHEMBL6205328

SCHEMBL6205328

CC(=O)Oc1cccc(CNc2nc(N(CCO)C(C)C)nc3nn[nH]c23)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
STAT3 P40763 2/20 0.36
PDE5A O76074 2/20 0.35
PDE4D Q08499 2/20 0.35
PDE6C P51160 1/20 0.35
CCNE2 O96020 5/20 0.34
CCNE1 P24864 5/20 0.34
CDK2 P24941 5/20 0.34
CDK1 P06493 3/20 0.34
CDK5 Q00535 2/20 0.34
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
AURKB Q96GD4 1/20 0.34
CCNT1 O60563 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
CCNH P51946 1/20 0.33
MNAT1 P51948 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203806 0.87 STAT3 (0.36) STAT3PDE5APDE4DPDE6CCCNE2
SCHEMBL6204605 0.85 TSHR (0.32) PDE5APDE4DPDE6CCCNE2CCNE1
SCHEMBL6205608 0.84 PARP1 (0.36) PARP1STAT3PDE5APDE4DPDE6C
SCHEMBL6201142 0.84 CDK1 (0.46) PDE5APDE4DPDE6CCCNE2CCNE1
SCHEMBL6202208 0.82 CDK1 (0.33) PDE5APDE4DPDE6CCCNE2CCNE1
SCHEMBL3445690 0.79 STAT3 (0.41) PARP1STAT3CCNE1CDK2CDK1
SCHEMBL3446443 0.79 CDK1 (0.45) PARP1STAT3CCNE2CCNE1CDK2
SCHEMBL6205622 0.79 CCNE2 (0.35) PARP1PDE5APDE4DPDE6CCCNE2
SCHEMBL3445494 0.79 STAT3 (0.40) PARP1STAT3CCNE2CCNE1CDK2
SCHEMBL6204524 0.78 CCNE2 (0.34) PDE5APDE4DPDE6CCCNE2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed