SCHEMBL6201142

SCHEMBL6201142

CC(C)N(CCO)c1nc(NCc2ccccc2)c2[nH]nnc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 10/20 0.46
CDK5 Q00535 3/20 0.46
CDK2 P24941 7/20 0.43
CCNE2 O96020 5/20 0.43
CCNE1 P24864 5/20 0.43
CCNB1 P14635 6/20 0.40
CSNK1D P48730 1/20 0.38
CLK2 P49760 1/20 0.38
DYRK1A Q13627 1/20 0.38
HIPK4 Q8NE63 1/20 0.38
SRPK1 Q96SB4 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
PDE4D Q08499 3/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE5A O76074 2/20 0.37
PDE6C P51160 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
CCNB2 O95067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203326 0.86 CDK2 (0.38) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6203806 0.86 STAT3 (0.36) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6204529 0.85 CCNE2 (0.44) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6205328 0.84 PARP1 (0.36) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6202208 0.84 CDK1 (0.33) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6204524 0.83 CCNE2 (0.34) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6203858 0.82 LMNA (0.35) CDK1CDK5CCNT1CDK9
SCHEMBL6204605 0.81 TSHR (0.32) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6202508 0.81 LCK (0.30) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6205469 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed