SCHEMBL6203326

SCHEMBL6203326

CC(C)N(CCO)c1nc(NCc2ccccc2N)c2[nH]nnc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 11/20 0.38
CCNE1 P24864 10/20 0.38
CCNE2 O96020 5/20 0.38
CDK5 Q00535 4/20 0.38
AURKA O14965 1/20 0.38
CCNT1 O60563 2/20 0.37
CDK7 P50613 2/20 0.37
CDK9 P50750 2/20 0.37
CCNH P51946 2/20 0.37
CDK5R1 Q15078 2/20 0.37
CDK1 P06493 2/20 0.34
ATM Q13315 1/20 0.31
SYK P43405 1/20 0.31
JAK2 O60674 2/20 0.31
JAK1 P23458 2/20 0.31
TYK2 P29597 2/20 0.31
JAK3 P52333 2/20 0.31
PDE5A O76074 1/20 0.30
PDE6C P51160 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201142 0.86 CDK1 (0.46) CDK2CCNE1CCNE2CDK5CCNT1
SCHEMBL6202208 0.86 CDK1 (0.33) CDK2CCNE1CCNE2CDK5CDK1
SCHEMBL6202508 0.85 LCK (0.30) CDK2CCNE1CCNE2CDK5CDK1
SCHEMBL6204605 0.84 TSHR (0.32) CDK2CCNE1CCNE2CDK5CDK1
SCHEMBL6203171 0.82 CCNE1 (0.37) CDK2CCNE1CCNE2CDK5AURKA
SCHEMBL6204524 0.81 CCNE2 (0.34) CDK2CCNE1CCNE2CDK5CCNT1
SCHEMBL6204274 0.81 CCR4 (0.33) CDK2CCNE1CCNE2
SCHEMBL6204529 0.80 CCNE2 (0.44) CDK2CCNE1CCNE2CDK5CDK5R1
SCHEMBL6203855 0.80 CCNE1 (0.34) CDK2CCNE1CCNE2CDK5CCNT1
SCHEMBL6203460 0.78 MTOR (0.32) CDK2CCNE1CCNE2CDK5CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed