SCHEMBL6202445

SCHEMBL6202445

O=C(Cc1ccc(Cl)cc1)c1ccc(F)cc1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.71
NPC1 O15118 3/20 0.71
L3MBTL1 Q9Y468 2/20 0.69
MAPT P10636 1/20 0.68
TP53 P04637 1/20 0.54
EGFR P00533 2/20 0.53
ERBB2 P04626 2/20 0.53
GSK3B P49841 2/20 0.52
POLB P06746 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
PTPN1 P18031 1/20 0.50
VNN1 O95497 1/20 0.49
KLK7 P49862 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8956384 1.00 RAB9A (0.71) RAB9ANPC1L3MBTL1MAPTTP53
SCHEMBL6201900 0.90 RAB9A (0.59) RAB9ANPC1L3MBTL1MAPTTP53
SCHEMBL1753283 0.90 RAB9A (0.85) RAB9ANPC1L3MBTL1MAPTGSK3B
SCHEMBL5725840 0.83 RAB9A (1.00) RAB9ANPC1L3MBTL1MAPTGSK3B
SCHEMBL1393818 0.83 L3MBTL1 (0.76) RAB9ANPC1L3MBTL1MAPTGSK3B
SCHEMBL10649146 0.83 RAB9A (1.00) RAB9ANPC1L3MBTL1MAPTGSK3B
SCHEMBL5724883 0.83 RAB9A (0.68) RAB9ANPC1L3MBTL1MAPTTP53
SCHEMBL7167952 0.83 SRD5A2 (0.62) RAB9ANPC1L3MBTL1MAPTPTPN1
SCHEMBL6202254 0.82 TP53 (0.59) RAB9ANPC1TP53GSK3BPOLB
SCHEMBL38657578 0.82 RAB9A (0.62) RAB9ANPC1L3MBTL1MAPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
US-5532374-A Method of preparation of bis-quinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1996-07-02 US disclosed