SCHEMBL6202254

SCHEMBL6202254

O=C(CCc1ccc(F)cc1)c1ccc(Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.59
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
GPR84 Q9NQS5 2/20 0.52
SLC5A1 P13866 1/20 0.51
SLC5A2 P31639 1/20 0.51
POLB P06746 1/20 0.51
DRD2 P14416 5/20 0.50
DRD4 P21917 3/20 0.50
DRD3 P35462 2/20 0.50
CNR1 P21554 1/20 0.50
HTR7 P34969 1/20 0.50
DRD1 P21728 1/20 0.50
DRD5 P21918 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HTR1A P08908 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL657632 1.00 TP53 (0.59) TP53NPC1RAB9AGPR84SLC5A1
SCHEMBL10559396 0.91 NPC1 (0.67) NPC1RAB9ASLC5A1SLC5A2HTR7
SCHEMBL11123550 0.91 GPR84 (0.59) NPC1RAB9AGPR84POLBMEN1
SCHEMBL11431321 0.84 NPC1 (0.69) TP53NPC1RAB9AGPR84SLC5A1
SCHEMBL27366629 0.83 RAB9A (0.70) NPC1RAB9AGPR84SLC5A1SLC5A2
SCHEMBL20262696 0.83 NPC1 (0.56) NPC1RAB9ASLC5A1SLC5A2DRD2
SCHEMBL6158144 0.83 NPC1 (0.56) NPC1RAB9ASLC5A1SLC5A2HTR7
SCHEMBL11612967 0.83 HTR7 (0.59) NPC1RAB9ASLC5A1SLC5A2HTR7
SCHEMBL3078714 0.82 L3MBTL1 (0.68) NPC1RAB9AGPR84MEN1KMT2A
SCHEMBL659281 0.82 NPC1 (0.59) NPC1RAB9ASLC5A1SLC5A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed