SCHEMBL6202754

SCHEMBL6202754

CCCN(CO)c1nc(NCc2ccccc2)c2nn[nH]c2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.43
CDK1 P06493 1/20 0.43
PRUNE1 Q86TP1 1/20 0.42
CCNE1 P24864 7/20 0.40
CDK2 P24941 7/20 0.40
CCNE2 O96020 6/20 0.40
CCNT1 O60563 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
CCNH P51946 1/20 0.38
CDK5R1 Q15078 1/20 0.38
PPARG P37231 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
CYP3A4 P08684 3/20 0.37
KDM4E B2RXH2 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203167 0.85 CCNE1 (0.41) CDK5CDK1PRUNE1CCNE1CDK2
SCHEMBL6203247 0.84 CCNE2 (0.43) CCNE1CDK2CCNE2CYP3A4MAPK1
SCHEMBL6202760 0.84 CDK1 (0.40) CDK5CDK1PRUNE1CCNE1CDK2
SCHEMBL6205602 0.83 PARP1 (0.37) PRUNE1CCNE1CDK2CCNE2PDE4A
SCHEMBL7013189 0.82 CDK1 (0.42) CDK5CDK1PRUNE1CCNE1CDK2
SCHEMBL6204126 0.80 SLC29A1 (0.32) PRUNE1SLC29A1
SCHEMBL6204808 0.78 PRUNE1 (0.37) CDK5CDK1PRUNE1CCNE1CDK2
SCHEMBL6203494 0.78 PRUNE1 (0.40) CDK5CDK1PRUNE1CCNE1CDK2
SCHEMBL6204714 0.78 SLC29A1 (0.32) PRUNE1SLC29A1
SCHEMBL6205408 0.76 PRUNE1 (0.35) CDK1PRUNE1MEN1KMT2ASLC29A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed