SCHEMBL6205602

SCHEMBL6205602

CCCN(CO)c1nc(NCc2cccc(OC(C)=O)c2)c2nn[nH]c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
PRUNE1 Q86TP1 1/20 0.37
SLC26A6 Q9BXS9 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AURKA O14965 3/20 0.34
RPS6KB1 P23443 3/20 0.34
CCNE2 O96020 2/20 0.34
CCNE1 P24864 2/20 0.34
CDK2 P24941 2/20 0.34
ACHE P22303 3/20 0.33
AURKB Q96GD4 1/20 0.33
CACNA2D1 P54289 1/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE3B Q13370 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205608 0.87 PARP1 (0.36) PARP1PRUNE1SLC26A6HTTSMN1; SMN2
SCHEMBL6202754 0.83 CDK5 (0.43) PRUNE1SMN1; SMN2CCNE2CCNE1CDK2
SCHEMBL3445269 0.78 CDK2 (0.49) SMN1; SMN2AURKACCNE2CCNE1CDK2
SCHEMBL6203167 0.76 CCNE1 (0.41) PRUNE1AURKACCNE2CCNE1CDK2
SCHEMBL3445688 0.76 CDK2 (0.42) PARP1SLC26A6AURKARPS6KB1CCNE1
SCHEMBL3446440 0.76 CDK1 (0.47) PARP1CCNE1CDK2MAPT
SCHEMBL3445488 0.76 PARP1 (0.38) PARP1SLC26A6AURKARPS6KB1CCNE2
SCHEMBL6203494 0.75 PRUNE1 (0.40) PRUNE1CCNE2CCNE1CDK2PDE4D
SCHEMBL3444310 0.73 CDK1 (0.55)
SCHEMBL6205408 0.73 PRUNE1 (0.35) PRUNE1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed