SCHEMBL6203097

SCHEMBL6203097

O=C(NNc1ccc(Cl)cc1)Oc1cnc2c(F)cccc2c1O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.44
GRM5 P41594 1/20 0.36
TRPA1 O75762 1/20 0.36
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PTGS2 P35354 2/20 0.35
ATM Q13315 1/20 0.34
ALDH1A1 P00352 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX12 P18054 1/20 0.34
CYP2C19 P33261 1/20 0.34
AURKA O14965 1/20 0.34
EIF4EBP1 Q13541 1/20 0.33
LMNA P02545 1/20 0.33
SCN9A Q15858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6198759 0.84 GAA (0.38) GAAFNTAFNTBPTGS2ATM
SCHEMBL6201873 0.84 TET2 (0.34) GAAFNTAFNTBPTGS2ATM
SCHEMBL6202705 0.84 GAA (0.36) GAAFNTAFNTBPTGS2ATM
SCHEMBL6200560 0.81 GAA (0.52) GAAGRM5PTGS2ALDH1A1CYP1A2
SCHEMBL6198854 0.68 EGLN1 (0.54) TRPA1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6204065 0.68 GAA (0.47) GAAPTGS2ALDH1A1CYP1A2CYP3A4
SCHEMBL6200932 0.65 GAA (0.41) GAAPTGS2ALDH1A1CYP1A2CYP3A4
SCHEMBL6198572 0.65 PTGS2 (0.44) GAAPTGS2ALDH1A1CYP1A2CYP3A4
SCHEMBL1504425 0.65 PTGS2 (0.58) GAAPTGS2ALDH1A1CYP1A2CYP3A4
SCHEMBL6198567 0.65 GAA (0.43) GAAPTGS2ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042295-B1 4-HYDROXYQUINOLINE-3-CARBOXAMIDES AND HYDRAZIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN CO LLC (US) 2005-09-07 EP claimed