SCHEMBL6203301

SCHEMBL6203301

CC[C@H]1CC[C@@H](C(=O)O)N1C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C.CC[C@H]1CC[C@@H](C(N)=O)N1C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.44
CTSL P07711 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
CTSB P07858 1/20 0.42
CAPN1 P07384 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 1/20 0.39
HRH2 P25021 2/20 0.38
HRH1 P35367 2/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
REN P00797 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ACE P12821 1/20 0.35
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203298 1.00 MAPK1 (0.44) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL27630344 0.96 MAPK1 (0.44) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL646244 0.96 MAPK1 (0.44) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL647656 0.95 CTSS (0.46) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL6203357 0.88 CTSK (0.43) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL646335 0.84 CTSL (0.44) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL646794 0.80 MAPK1 (0.47) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL27611195 0.80 MAPK1 (0.47) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL6761081 0.80 MAPK1 (0.47) MAPK1CTSLCTSSCTSKCTSB
SCHEMBL14216709 0.79 CTSK (0.44) CTSLCTSSCTSKCTSBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560811-A2 PHARMACEUTICAL COMPOSITIONS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-IV) Abbott Laboratories (US) 2005-08-10 EP disclosed
WO-2004026822-A2 PHARMACEUTICAL COMPOSITIONS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-IV) ABBOTT LABORATORIES (US) 2004-04-01 WO disclosed