SCHEMBL6203419

SCHEMBL6203419

Cc1ccc(C(=O)NC(=O)[C@H]2CCCCN2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
GABRA5 P31644 3/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
KDM4E B2RXH2 1/20 0.42
WNT1 P04628 1/20 0.40
GSK3B P49841 1/20 0.40
DYRK1A Q13627 1/20 0.40
KMT2A Q03164 1/20 0.40
PRKAB2 O43741 1/20 0.39
PRKAG1 P54619 1/20 0.39
PRKAA2 P54646 1/20 0.39
PRKAA1 Q13131 1/20 0.39
PRKAG3 Q9UGI9 1/20 0.39
PRKAG2 Q9UGJ0 1/20 0.39
PRKAB1 Q9Y478 1/20 0.39
ULK1 O75385 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6265321 0.82 HPGD (0.42) NPC1ALDH1A1MAPTKDM4EWNT1
SCHEMBL20037446 0.79 ULK1 (0.54) WNT1GSK3BDYRK1AULK1SCN3A
SCHEMBL6277414 0.79 SMYD3 (0.47) NPC1ALDH1A1WNT1GSK3BDYRK1A
SCHEMBL8727230 0.78 GSK3B (0.38) WNT1GSK3BDYRK1ASCN3ASCN9A
SCHEMBL14490487 0.78 HTT (0.53) HDAC1HDAC6ALDH1A1MAPT
SCHEMBL6204321 0.76 HDAC1 (0.48) HDAC1HDAC6WNT1GSK3BDYRK1A
SCHEMBL6203532 0.76 HDAC1 (0.48) HDAC1HDAC6WNT1GSK3BDYRK1A
SCHEMBL6203499 0.76 HDAC1 (0.48) HDAC1HDAC6WNT1GSK3BDYRK1A
SCHEMBL6371533 0.75 HDAC1 (0.50) HDAC1HDAC6NPC1ALDH1A1MAPT
SCHEMBL8397188 0.74 CTSC (0.49) HDAC1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed