SCHEMBL6203499

SCHEMBL6203499

Cc1ccc(C(=O)NC(=O)[C@H]2CCCNC2)cn1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
WNT1 P04628 2/20 0.41
GSK3B P49841 2/20 0.41
DYRK1A Q13627 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204321 1.00 HDAC1 (0.48) HDAC1HDAC6WNT1GSK3BDYRK1A
SCHEMBL6203532 1.00 HDAC1 (0.48) HDAC1HDAC6WNT1GSK3BDYRK1A
SCHEMBL6371533 0.92 HDAC1 (0.50) HDAC1HDAC6
SCHEMBL6204294 0.82 ALDH1A1 (0.51) HDAC1HDAC6
SCHEMBL3879671 0.79 NPC1 (0.47)
SCHEMBL6203700 0.79 KDM4E (0.45)
SCHEMBL6204513 0.79 SMYD3 (0.46) WNT1GSK3BDYRK1A
SCHEMBL6204397 0.79 SMYD3 (0.46) WNT1GSK3BDYRK1A
SCHEMBL1996065 0.76
SCHEMBL1996068 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed