SCHEMBL6203460

SCHEMBL6203460

COc1cc(O)c(CNc2nc(N(CCO)C(C)C)nc3nn[nH]c23)cc1O

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.32
CDK1 P06493 3/20 0.32
CCNB1 P14635 3/20 0.32
PDE5A O76074 2/20 0.32
PDE4D Q08499 2/20 0.32
CCNB2 O95067 2/20 0.32
CCNB3 Q8WWL7 2/20 0.32
PDE6C P51160 1/20 0.32
CCNT1 O60563 1/20 0.32
CCNE2 O96020 1/20 0.32
CCNA2 P20248 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
CCNH P51946 1/20 0.32
MNAT1 P51948 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203855 0.86 CCNE1 (0.34) MTORCDK1CCNB1PDE5APDE4D
SCHEMBL6205414 0.83 HMGCR (0.32) PRUNE1
SCHEMBL6205469 0.81
SCHEMBL6204274 0.78 CCR4 (0.33) CCNE2CCNE1CDK2
SCHEMBL6203326 0.78 CDK2 (0.38) CDK1CCNB1PDE5APDE4DCCNB2
SCHEMBL3444371 0.78 CDK2 (0.36) CDK1CCNB1CCNB2CCNB3CCNT1
SCHEMBL3445346 0.78 CDK1 (0.41) CDK1CCNB1CCNB2CCNB3CCNT1
SCHEMBL6204605 0.77 TSHR (0.32) CDK1PDE5APDE4DPDE6CCCNE2
SCHEMBL6201142 0.77 CDK1 (0.46) CDK1CCNB1PDE5APDE4DCCNB2
SCHEMBL3445020 0.77 SYK (0.35) CDK1CCNB1CCNB2CCNB3CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed