SCHEMBL6204448

SCHEMBL6204448

O=C1[N]c2cc(Nc3ccccc3)c(Cc3cccc(Cl)c3Cl)cc2N1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GSK3B P49841 2/20 0.34
MAPK1 P28482 2/20 0.34
LMNA P02545 2/20 0.34
ALDH1A1 P00352 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
KDM4E B2RXH2 1/20 0.34
RGS12 O14924 1/20 0.34
GMNN O75496 1/20 0.34
PRKD3 O94806 1/20 0.34
EGFR P00533 1/20 0.34
PRKCG P05129 1/20 0.34
PRKCB P05771 1/20 0.34
GLA P06280 1/20 0.34
CYP3A4 P08684 1/20 0.34
SRC P12931 1/20 0.34
HPGD P15428 1/20 0.34
PRKCA P17252 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204202 0.85 CXCR2 (0.36) MAPTMEN1KMT2AGSK3BMAPK1
SCHEMBL6205665 0.83 EGFR (0.36) MAPTMEN1KMT2AMAPK1LMNA
SCHEMBL6203291 0.83 EGFR (0.39) MAPTMEN1KMT2AMAPK1LMNA
SCHEMBL6205378 0.83 KMT2A (0.40) MAPTMEN1KMT2AGSK3BMAPK1
SCHEMBL6205452 0.83 EGFR (0.36) MAPTMEN1KMT2AGSK3BMAPK1
SCHEMBL6204330 0.82 CNR1 (0.39) MAPTMEN1KMT2AGSK3BMAPK1
SCHEMBL6202957 0.82 ALDH1A1 (0.35) MAPTMEN1KMT2AGSK3BMAPK1
SCHEMBL6204309 0.78 RAB9A (0.40) MAPTMEN1KMT2AMAPK1LMNA
SCHEMBL6203101 0.78 NPC1 (0.38) MAPTMEN1KMT2AGSK3BMAPK1
SCHEMBL6205611 0.77 MEN1 (0.38) MAPTMEN1KMT2AMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539708-A1 BENZIMIDAZOLONES AND THEIR USE AS CYTOKINE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2005-06-15 EP disclosed
WO-2004024699-A1 BENZIMIDAZOLONES AND THEIR USE AS CYTOKINE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2004-03-25 WO disclosed