SCHEMBL6204543

SCHEMBL6204543

CCCN(CO)c1nc(NCc2ccccc2N)c2c(n1)N(C(C)C)NN2C(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 8/20 0.37
CDK2 P24941 8/20 0.37
CDK5 Q00535 4/20 0.37
CCNE2 O96020 3/20 0.37
AURKA O14965 1/20 0.37
CCNT1 O60563 2/20 0.35
CDK7 P50613 2/20 0.35
CDK9 P50750 2/20 0.35
CCNH P51946 2/20 0.35
CDK5R1 Q15078 2/20 0.35
CDK1 P06493 1/20 0.33
PDE5A O76074 1/20 0.30
PDE6C P51160 1/20 0.30
PDE4D Q08499 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205006 0.87 CDK1 (0.44) CCNE1CDK2CDK5CCNE2CCNT1
SCHEMBL6204991 0.84 PKM (0.42) CCNE1CDK2CCNE2CCNT1CDK9
SCHEMBL6203902 0.82 CCNE2 (0.31) CCNE1CDK2CCNE2
SCHEMBL6205631 0.81 CCNE2 (0.44) CCNE1CDK2CDK5CCNE2CDK5R1
SCHEMBL6204092 0.80 CCNT1 (0.31) CCNE1CDK2CDK5CCNT1CDK7
SCHEMBL6205415 0.78 CDK1 (0.34) CCNE1CDK2CDK5CCNE2CCNT1
SCHEMBL3446046 0.78 CDK1 (0.48) CCNE1CDK2CDK5CCNE2AURKA
SCHEMBL3446768 0.77 CDK2 (0.60) CCNE1CDK2CDK5CCNE2AURKA
SCHEMBL6204186 0.77 PDE5A (0.36) CCNE1CDK2CDK5CCNE2CCNT1
SCHEMBL3444119 0.76 CDK2 (0.57) CCNE1CDK2CDK5CCNE2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed