SCHEMBL6205631

SCHEMBL6205631

CCCN(CO)c1nc(Nc2ccccc2)c2c(n1)N(C(C)C)NN2C(C)C

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 5/20 0.44
CCNE1 P24864 5/20 0.44
CDK2 P24941 5/20 0.44
ADORA2A P29274 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
CDK5 Q00535 2/20 0.33
ATM Q13315 1/20 0.33
CDK5R1 Q15078 1/20 0.33
HTR2C P28335 3/20 0.32
CDK1 P06493 1/20 0.32
HTR2A P28223 1/20 0.31
KCNH3 Q9ULD8 3/20 0.31
CFTR P13569 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206198 0.90 CCNE2 (0.46) CCNE2CCNE1CDK2HTR2CCDK1
SCHEMBL6203776 0.89 CDK5 (0.46) CCNE2CCNE1CDK2CDK5ATM
SCHEMBL6205006 0.86 CDK1 (0.44) CCNE2CCNE1CDK2CDK5CDK5R1
SCHEMBL6203210 0.83 CCNE2 (0.42) CCNE2CCNE1CDK2CDK5ATM
SCHEMBL6204543 0.81 CCNE1 (0.37) CCNE2CCNE1CDK2CDK5CDK5R1
SCHEMBL6203902 0.76 CCNE2 (0.31) CCNE2CCNE1CDK2
SCHEMBL6205415 0.76 CDK1 (0.34) CCNE2CCNE1CDK2CDK5CDK5R1
SCHEMBL6204991 0.76 PKM (0.42) CCNE2CCNE1CDK2
SCHEMBL3445689 0.75 CDK5 (0.46) CCNE2CCNE1CDK2CDK5CDK5R1
SCHEMBL3445478 0.74 KCNH3 (0.53) CCNE2CCNE1CDK2CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed