SCHEMBL6205415

SCHEMBL6205415

CCCN(CO)c1nc(NCc2cccc(C(C)=O)c2)c2c(n1)N(C(C)C)NN2C(C)C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.34
CDK5 Q00535 2/20 0.34
CCNE2 O96020 7/20 0.33
CCNE1 P24864 7/20 0.33
CDK2 P24941 7/20 0.33
PDE5A O76074 3/20 0.32
PDE4D Q08499 3/20 0.32
PDE6C P51160 2/20 0.32
TRPV3 Q8NET8 1/20 0.32
WDR5 P61964 1/20 0.31
CTNNB1 P35222 1/20 0.31
TCF7L2 Q9NQB0 1/20 0.31
JAK3 P52333 1/20 0.30
STAT3 P40763 1/20 0.30
CCNT1 O60563 1/20 0.30
CCNB1 P14635 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK7 P50613 1/20 0.30
CDK9 P50750 1/20 0.30
CCNH P51946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205006 0.87 CDK1 (0.44) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6203737 0.86 CDK1 (0.36) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL3444723 0.80 CDK1 (0.47) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL3444325 0.79 CDK2 (0.50) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL3443903 0.78 CDK2 (0.42) CDK1CDK5CCNE1CDK2JAK3
SCHEMBL6204543 0.78 CCNE1 (0.37) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL3444183 0.78 BCDIN3D (0.39) CDK1CCNE2CCNE1CDK2STAT3
SCHEMBL6204991 0.77 PKM (0.42) CCNE2CCNE1CDK2CCNT1CDK9
SCHEMBL6205631 0.76 CCNE2 (0.44) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6204092 0.75 CCNT1 (0.31) CDK5CCNE1CDK2CCNT1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed